TOLPERITAS 150 TABLET

🦴💊🧘 Tolperisone 150mg Tablet: Advanced Muscle Relaxant for Spasticity & Pain Relief

Tolperisone 150mg is a centrally acting muscle relaxant widely used for the treatment of muscle spasticity, muscle stiffness, and neurological conditions that cause increased muscle tone. It is particularly effective in neuromuscular disorders, spinal cord diseases, and post-stroke muscle tightness, offering both muscle relaxation and pain relief without significant sedation.

As a higher strength formulation, Tolperisone 150mg is suitable for moderate to severe muscle spasms or when lower doses are insufficient. It improves mobility, reduces discomfort, and enhances the quality of life in patients suffering from muscular and neurological disorders.

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🔬 Mechanism of Action

Tolperisone acts on the central nervous system (CNS) to:

• Block voltage-gated sodium and calcium channels in nerve cells

• Inhibit excessive nerve impulses that cause muscle spasticity

• Reduce muscle stiffness without causing drowsiness or loss of motor coordination

• Improve blood circulation in muscle tissues by relaxing vascular smooth muscles

This dual neuromuscular and vasodilatory action makes it beneficial for both muscle-related pain and circulatory disorders associated with muscle spasticity.

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📌 Indications and Uses

Tolperisone 150mg is prescribed for:

• Spasticity due to neurological conditions like stroke, multiple sclerosis, and spinal cord injury

• Muscle spasms associated with degenerative vertebral diseases (e.g., cervical or lumbar spondylosis)

• Post-operative muscle stiffness

• Muscle rigidity in conditions like cerebral palsy or Parkinson’s disease (as adjunct)

• Peripheral vascular diseases with associated muscle cramps (in select cases)

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💊 Dosage and Administration

• Standard dose: 150mg two to three times daily after meals

• Dosage should be individualized based on patient’s condition, severity of spasticity, and tolerability

• Swallow tablet whole, do not crush or chew

Note: Tolperisone should always be taken with food to improve absorption and reduce gastrointestinal side effects.

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⚠️ Precautions and Warnings

• Not suitable for:

  • Children under 18 years

  • Patients with myasthenia gravis (muscle weakness disorder)

  • Known hypersensitivity to tolperisone or any inactive ingredients

• Use with caution in:

  • Liver or kidney impairment

  • Pregnant or breastfeeding women (only if clearly needed)

  • Elderly patients

Driving or operating machinery is generally safe, but caution is advised until individual response is known.

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🤒 Side Effects

Common:

• Headache

• Dizziness

• Nausea

• Fatigue

• Abdominal discomfort

Rare/Serious:

• Allergic reactions: rash, itching, swelling

• Hypotension (low blood pressure)

• Muscle weakness or coordination issues (uncommon)

Discontinue immediately if signs of allergy or severe adverse effects occur.

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🔄 Drug Interactions

• Use caution with:

  • CNS depressants (e.g., benzodiazepines, alcohol)

  • Muscle relaxants or antihypertensive medications

• Limited known interactions, but inform the doctor about all ongoing medications

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🧊 Storage Instructions

• Store below 25°C, away from moisture and direct sunlight

• Keep out of reach of children

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📝 Conclusion

Tolperisone 150mg is a well-tolerated, non-sedative muscle relaxant that effectively treats spasticity, stiffness, and muscle pain across a range of neuromuscular disorders. Its unique ability to relieve muscular symptoms without impairing alertness makes it a preferred choice for patients needing long-term relief and improved physical function. Always use under medical supervision for optimal results.

Note: This information is intended for educational purposes and should not replace professional medical advice. Always consult a healthcare provider for personalized guidance.